SCHEMBL5048859

SCHEMBL5048859

CCCn1c(=O)c2c(nc(CC(=O)c3nscc3F)n2CCN(CC)CCO)n(CCc2ccccc2N)c1=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.43
TSHR P16473 4/20 0.35
ADORA2B P29275 6/20 0.33
ADORA2A P29274 3/20 0.33
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.30
JAK2 O60674 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1333093 0.88 ADORA1 (0.45) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL1334380 0.84 ADORA1 (0.53) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL4167641 0.81 ADORA1 (0.52) ADORA1TSHRADORA2BADORA2ALMNA
Hydrochloric Acid SCHEMBL4174153 0.80 ADORA1 (0.51) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL1333068 0.80 ADORA1 (0.48) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL4182302 0.80 ADORA1 (0.59) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL1332421 0.78 ADORA1 (0.40) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL1333058 0.77 ADORA1 (0.48) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL1333442 0.77 ADORA1 (0.46) ADORA1TSHRADORA2BADORA2ALMNA
SCHEMBL2073738 0.77 ADORA1 (0.48) ADORA1TSHRADORA2BADORA2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636229-A4 A1 ADENOSINE RECEPTOR ANTOGONISTS ENDACEA INC (US) 2008-07-30 EP disclosed
EP-1636229-A2 A1 ADENOSINE RECEPTOR ANTOGONISTS Endacea, Inc. (US) 2006-03-22 EP disclosed
WO-2005009343-A2 A1 ADENOSINE RECEPTOR ANTOGONISTS ENDACEA, INC. (US) 2005-02-03 WO disclosed