SCHEMBL5048992

SCHEMBL5048992

CCCCCCCCCCCc1noc(-c2ccc(C([N][O])[C@H](C)c3ccc(C(F)(F)F)cc3)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
SPHK1 Q9NYA1 1/20 0.39
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
S1PR1 P21453 1/20 0.36
ADORA2B P29275 4/20 0.36
ADORA1 P30542 2/20 0.36
ADORA2A P29274 1/20 0.36
SPHK2 Q9NRA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5045551 1.00 KDM4E (0.39) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL5047608 1.00 KDM4E (0.39) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL5045607 0.81 NPC1 (0.41) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL5039728 0.80 PPARG (0.41) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL5039579 0.80 PPARG (0.41) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL5048708 0.80 PPARG (0.41) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL1857189 0.79 SPHK1 (0.46) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL1856616 0.79 SPHK1 (0.46) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL1856411 0.79 SPHK1 (0.46) KDM4ENPC1ALDH1A1MAPTPKM
SCHEMBL6783418 0.79 NPC1 (0.47) KDM4ENPC1ALDH1A1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed