SCHEMBL5050595

SCHEMBL5050595

CC(C)(C)OC(=O)N1CCN(C(=O)c2ccc3c(c2)cc(-c2ccc(-c4cccs4)c4c2C(=O)NC4)n3C(=O)OC(C)(C)C)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.40
GPR119 Q8TDV5 2/20 0.39
CNR2 P34972 1/20 0.38
LTK P29376 1/20 0.37
CDK5 Q00535 1/20 0.37
MST1R Q04912 1/20 0.37
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
ABL1 P00519 4/20 0.37
BCR P11274 4/20 0.37
CRBN Q96SW2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
AKT1 P31749 1/20 0.34
DYRK2 Q92630 1/20 0.34
HDAC4 P56524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3034098 0.88 CRBN (0.41) GBA1CNR2CRBNMEN1KMT2A
SCHEMBL3039265 0.87 MEN1 (0.41) GPR119CNR2CRBNMEN1KMT2A
SCHEMBL3041591 0.87 MEN1 (0.43) GPR119CNR2CRBNMEN1KMT2A
SCHEMBL3050148 0.86 CFTR (0.39) GPR119CNR2CRBNMEN1KMT2A
SCHEMBL3044424 0.86 CACNA1B (0.39) GPR119CNR2CRBNMEN1KMT2A
SCHEMBL3151651 0.84 MEN1 (0.36) GPR119CNR2CRBNMEN1KMT2A
SCHEMBL3046089 0.84 CCNA2 (0.40) CNR2CRBNMEN1KMT2ANR1H2
SCHEMBL3047862 0.83 GBA1 (0.39) GBA1GPR119CNR2ABL1BCR
SCHEMBL3048669 0.82 LTK (0.36) LTKCDK5MST1RDYRK1ACLK4
SCHEMBL3033984 0.80 MEN1 (0.43) GPR119CNR2CRBNMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed