SCHEMBL5050602

SCHEMBL5050602

COc1cc(-c2cc3cc(CNCCN(C)C)ccc3n2C(=O)OC(C)(C)C)c2c(c1OS(C)(=O)=O)CNC2=O

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.34
ATR Q13535 1/20 0.31
ATRIP Q8WXE1 1/20 0.31
NQO2 P16083 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3051282 0.96 NR1H2 (0.33) NR1H2ATRATRIP
SCHEMBL3043909 0.93 NR1H2 (0.35) NR1H2NQO2NR1H3
SCHEMBL3046270 0.92 NR1H2 (0.34) NR1H2NQO2NR1H3
SCHEMBL3049037 0.91 NR1H2 (0.36) NR1H2NQO2NR1H3
SCHEMBL3047918 0.91 NR1H2 (0.32) NR1H2
SCHEMBL3039682 0.91 NR1H2 (0.33) NR1H2
SCHEMBL3034109 0.91 NR1H2 (0.34) NR1H2ATRATRIPNQO2
SCHEMBL3040869 0.91 NR1H2 (0.41) NR1H2NR1H3
SCHEMBL3049654 0.90 NR1H2 (0.36) NR1H2ATRATRIPNQO2NR1H3
SCHEMBL3047552 0.90 NR1H2 (0.36) NR1H2NQO2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed