SCHEMBL5060263

SCHEMBL5060263

CC(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc(-c4cn[nH]c4)c3)cc2)n(-c2ccc3[nH]cnc3c2)n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.47
KDR P35968 9/20 0.44
ABL1 P00519 3/20 0.42
AXL P30530 2/20 0.42
FLT3 P36888 1/20 0.41
MAPK14 Q16539 2/20 0.41
MAPK13 O15264 2/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
KCNJ6 P48051 1/20 0.41
KCNJ5 P48544 1/20 0.41
KCNJ3 P48549 1/20 0.41
SRC P12931 2/20 0.41
RAF1 P04049 1/20 0.40
FLT1 P17948 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5052148 0.91 MAPK14 (0.44) BRAFKDRABL1AXLFLT3
SCHEMBL5052992 0.89 ABL1 (0.56) BRAFABL1AXLFLT3MAPK14
SCHEMBL5060321 0.88 BRAF (0.47) BRAFKDRABL1AXLFLT3
SCHEMBL5055072 0.88 MAPK14 (0.48) BRAFKDRABL1AXLFLT3
SCHEMBL5060252 0.86 ABL1 (0.59) BRAFKDRABL1AXLFLT3
SCHEMBL5054974 0.86 BRAF (0.49) BRAFKDRABL1AXLFLT3
SCHEMBL5056409 0.86 ABL1 (0.57) BRAFKDRABL1AXLFLT3
SCHEMBL5056317 0.85 BRAF (0.50) BRAFKDRAXLFLT3MAPK14
SCHEMBL5054691 0.85 KCNJ6 (0.52) BRAFKDRAXLMAPK14MAPK13
SCHEMBL5052280 0.85 BRAF (0.49) BRAFABL1AXLFLT3MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080113967-A1 ENZYME MODULATORS AND TREATMENTS DECIPHERA PHARMACEUTICALS, LLC (US) 2008-05-15 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080113967-A1 ENZYME MODULATORS AND TREATMENTS ABL2, BRAF, MAP3K1 BRAF 2/4885KDR 41/4885ABL1 20/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.