SCHEMBL5067541

SCHEMBL5067541

O=S(=O)(NCC1CCC(OCCCCCCN2CC=CCC2)CC1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.40
KCNH2 Q12809 1/20 0.40
HTR7 P34969 5/20 0.40
USP30 Q70CQ3 1/20 0.39
CCR1 P32246 1/20 0.39
HTR1A P08908 3/20 0.38
DRD2 P14416 3/20 0.38
HTR6 P50406 3/20 0.38
TGFBR1 P36897 1/20 0.37
MGLL Q99685 1/20 0.36
EPHX2 P34913 2/20 0.36
GBA1 P04062 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
GLA P06280 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065682 0.88 HRH3 (0.49) HRH3KCNH2HTR7USP30CCR1
SCHEMBL5088018 0.84 HRH3 (0.42) HRH3KCNH2HTR7USP30CCR1
SCHEMBL4806286 0.81 HTR2A (0.52) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL4806291 0.81 HTR2A (0.52) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL4806191 0.80 HTR2A (0.53) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL4806187 0.80 HTR2A (0.53) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL4799025 0.78 HTR2A (0.53) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL4799028 0.78 HTR2A (0.53) HRH3HTR7HTR1ADRD2ALDH1A1
SCHEMBL7204735 0.77 CA1 (0.43) TGFBR1GBA1HPGDHTTALDH1A1
SCHEMBL7211522 0.77 USP30 (0.44) USP30TGFBR1MGLLGBA1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311475-B1 AMINOCYCLOHEXANE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-08-06 EP disclosed