SCHEMBL5067647

SCHEMBL5067647

O=C(NCC1(F)CCN(C(=O)O)CC1)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.64
SCN5A Q14524 1/20 0.54
CACNA1I Q9P0X4 1/20 0.54
P2RX7 Q99572 1/20 0.48
SMYD3 Q9H7B4 1/20 0.44
CACNA1H O95180 2/20 0.43
CYP2D6 P10635 2/20 0.43
FABP4 P15090 1/20 0.43
CCKBR P32239 2/20 0.42
HTR1A P08908 2/20 0.42
RAB9A P51151 1/20 0.41
CHRNA7 P36544 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2889178 0.83 KCNH2 (0.73) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2886502 0.82 KCNH2 (0.65) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2887799 0.82 KCNH2 (0.79) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2889566 0.80 KCNH2 (0.79) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2885705 0.80 KCNH2 (0.73) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2881952 0.80 KCNH2 (0.69) KCNH2SCN5ACACNA1IP2RX7SMYD3
SCHEMBL2885274 0.80 KCNH2 (0.59) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2881082 0.79 KCNH2 (0.74) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL2886760 0.79 KCNH2 (0.64) KCNH2SCN5ACACNA1IP2RX7CACNA1H
SCHEMBL14693995 0.78 KCNH2 (0.44) KCNH2SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1901746-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2008-03-26 EP disclosed
WO-2007002884-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-01-04 WO disclosed