SCHEMBL506803

SCHEMBL506803

CC(C)(C)c1nc(N(C(=O)O)C(C)(C)C)c(-c2cc(-c3ccc(CNC4CC4)cc3)no2)nc1-c1ccc(=O)[nH]c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATR Q13535 9/20 0.44
PRKD1 Q15139 6/20 0.40
ATM Q13315 1/20 0.38
PRKD3 O94806 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16205157 0.80 PRKD1 (0.46) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL16205734 0.77 PRKD1 (0.45) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL506069 0.74 PRKD1 (0.42) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL2636029 0.74 ATR (0.57) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL506783 0.73 PPARA (0.35) ATRATM
SCHEMBL506949 0.73 PPARA (0.35) ATRATM
SCHEMBL10178131 0.72 ATR (0.54) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL506447 0.72 ATR (0.77) ATRATM
SCHEMBL12988352 0.68 ATR (0.44) ATRPRKD1ATMPRKD3PRKD2
SCHEMBL14859933 0.67 ATR (0.43) ATRPRKD1ATMPRKD3PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9630956-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-04-25 US disclosed
US-20120027874-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120027874-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, CHEK2 ATR 1/4885PRKD1 89/4885ATM 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.