SCHEMBL5069851

SCHEMBL5069851

COc1cc(OC)cc(C(=O)NCC2(C(F)C(=O)N3CCCC3C(F)(F)F)CCNCC2)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
KCNH2 Q12809 11/20 0.41
CACNA1G O43497 2/20 0.41
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.38
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPT P10636 1/20 0.37
GAA P10253 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PREP P48147 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5071693 0.94 NPC1 (0.39) NPC1KCNH2CACNA1GALDH1A1POLB
SCHEMBL5069860 0.87 KCNH2 (0.41) KCNH2CACNA1G
SCHEMBL5069843 0.84 CACNA1H (0.40) KCNH2CACNA1G
SCHEMBL2886010 0.76 NPC1 (0.46) NPC1KCNH2CACNA1GTSHRMAPT
SCHEMBL2890369 0.71 KCNH2 (0.50) NPC1KCNH2CACNA1G
SCHEMBL4274547 0.70 KMT2A (0.47) NPC1KCNH2CACNA1GALDH1A1POLB
SCHEMBL4274552 0.70 KMT2A (0.47) NPC1KCNH2CACNA1GALDH1A1POLB
SCHEMBL14708779 0.70 NPC1 (0.53) NPC1KCNH2CACNA1GTSHRHPGD
SCHEMBL4279685 0.66 CACNA1I (0.49) NPC1KCNH2CACNA1GALDH1A1POLB
SCHEMBL4270883 0.66 CACNA1I (0.49) NPC1KCNH2CACNA1GALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1901746-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2008-03-26 EP claimed
WO-2007002884-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-01-04 WO claimed