SCHEMBL5080339

SCHEMBL5080339

CN(C)CCOc1ccc(C(=C(c2ccc(O)cc2)C(F)(F)F)c2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.70
ESRRG P62508 12/20 0.67
ESRRB O95718 6/20 0.67
ESR2 Q92731 4/20 0.67
MAPT P10636 3/20 0.67
MEN1 O00255 2/20 0.67
TP53 P04637 2/20 0.67
CYP3A4 P08684 2/20 0.67
KMT2A Q03164 2/20 0.67
PGR P06401 2/20 0.67
KDM4E B2RXH2 1/20 0.67
ALDH1A1 P00352 1/20 0.67
LMNA P02545 1/20 0.67
HIF1A Q16665 1/20 0.67
NPSR1 Q6W5P4 1/20 0.67
PLD2 O14939 1/20 0.67
PLD1 Q13393 1/20 0.67
ESRRA P11474 3/20 0.62
NPC1 O15118 1/20 0.58
NR1I2 O75469 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10484358 1.00 ESR1 (0.70) ESR1ESRRGESRRBESR2MAPT
SCHEMBL1151837 1.00 ESR1 (0.70) ESR1ESRRGESRRBESR2MAPT
SCHEMBL10484026 1.00 ESR1 (0.70) ESR1ESRRGESRRBESR2MAPT
Hydrochloric Acid SCHEMBL10484008 0.99 ESR1 (0.68) ESR1ESRRGESRRBESR2MAPT
Hydrochloric Acid SCHEMBL10484012 0.99 ESR1 (0.68) ESR1ESRRGESRRBESR2MAPT
SCHEMBL1152006 0.95 ESR1 (0.61) ESR1ESRRGESRRBESR2MAPT
SCHEMBL1152003 0.95 ESR1 (0.61) ESR1ESRRGESRRBESR2MAPT
SCHEMBL10484027 0.95 ESR1 (0.64) ESR1ESRRGESRRBESR2MAPT
SCHEMBL10484033 0.95 ESR1 (0.64) ESR1ESRRGESRRBESR2MAPT
SCHEMBL10484030 0.95 ESR1 (0.64) ESR1ESRRGESRRBESR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008133884-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-11-06 WO disclosed
US-4806685-A EXERTS VARIOUS EFFECTS ON ENDOCRINOUS SYSTEM OF RATS; INHIBITS GROWTH OF MAMMARY TUMORS GYOGYSZERKUTATO INTEEZET/PHARMACEUTICAL RESEARCH INSTITUTE (HU) 1989-02-21 US disclosed