SCHEMBL5082092

SCHEMBL5082092

O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2Cc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 20/20 0.83
HDAC8 Q9BY41 16/20 0.83
HDAC2 Q92769 15/20 0.83
HDAC1 Q13547 4/20 0.48
HDAC3 O15379 2/20 0.47
HDAC4 P56524 2/20 0.47
HDAC7 Q8WUI4 2/20 0.47
HDAC10 Q969S8 2/20 0.47
HDAC11 Q96DB2 2/20 0.47
HDAC9 Q9UKV0 2/20 0.47
HDAC5 Q9UQL6 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5075672 0.92 HDAC6 (0.76) HDAC6HDAC8HDAC2HDAC1HDAC3
SCHEMBL5075670 0.92 HDAC6 (0.76) HDAC6HDAC8HDAC2HDAC1HDAC3
SCHEMBL5078399 0.91 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5078396 0.91 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5082166 0.91 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5579314 0.90 HDAC6 (0.86) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5078349 0.90 HDAC6 (0.86) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5078389 0.89 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5078392 0.89 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1
SCHEMBL5077642 0.85 HDAC6 (1.00) HDAC6HDAC8HDAC2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101296910-A Benzodiazepine and benzopiperazine analog inhibitors of histone deacetylase METHYLGENE INC (CA) 2008-10-29 CN claimed
EP-1940805-A1 BENZODIAZEPINE AND BENZOPIPERAZINE ANALOG INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2008-07-09 EP claimed
WO-2007022638-A1 BENZODIAZEPINE AND BENZOPIPERAZINE ANALOG INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2007-03-01 WO claimed
CN-101296910-A Benzodiazepine and benzopiperazine analog inhibitors of histone deacetylase METHYLGENE INC (CA) 2008-10-29 CN disclosed