Bromide

Bromide

SCHEMBL5084016

Br.Br.c1ccc2sc(SCCCCCCSc3nc4ccccc4s3)nc2c1

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 1/20 0.65
ADRA2A known ✓ P08913 1/20 0.59
ADRA2B known ✓ P18089 1/20 0.59
ADRA2C known ✓ P18825 1/20 0.59
SLC6A3 known ✓ Q01959 1/20 0.59
CYP1A2 P05177 4/20 0.80
CYP2D6 P10635 3/20 0.80
CYP2C19 P33261 3/20 0.71
CYP3A4 P08684 2/20 0.71
CYP2C9 P11712 1/20 0.71
STAT6 P42226 1/20 0.71
MAPK1 P28482 2/20 0.69
HIF1A Q16665 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
ALDH1A1 P00352 6/20 0.68
SMN1; SMN2 Q16637 5/20 0.68
KDM4E B2RXH2 2/20 0.68
GFER P55789 1/20 0.68
HTR2A P28223 1/20 0.65
HTR7 P34969 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141647 0.98 CYP1A2 (0.83) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL19614388 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL2208304 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL11590344 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL7401382 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL15501213 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL30423175 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL11299646 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL11339285 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL12371907 0.91 CYP1A2 (0.71) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7358313-B2 Thiouronium salt as anti-reversion agent in a vulcanizable rubber composition and tire based on such a composition MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-04-15 US disclosed
US-20050187340-A1 Thiouronium salt as anti-reversion agent in a vulcanizable rubber composition and tire based on such a composition MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2005-08-25 US disclosed