SCHEMBL5084730

SCHEMBL5084730

Cc1cc(N2CCC[C@H]2CO)c2ccc(N)cc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.42
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
NQO2 P16083 2/20 0.40
ACVR1 Q04771 2/20 0.40
MAP2K7 O14733 1/20 0.39
NCF1 P14598 3/20 0.38
PDK2 Q15119 2/20 0.38
PDK4 Q16654 1/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
NR1I2 O75469 1/20 0.38
SMARCA2 P51531 1/20 0.38
SMARCA4 P51532 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
PBRM1 Q86U86 1/20 0.38
ADORA2A P29274 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025400 1.00 CCNE2 (0.42) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5036104 0.87 MAP2K7 (0.48) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5036101 0.87 MAP2K7 (0.48) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5022604 0.86 ADORA2A (0.46) NQO2ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5091471 0.86 ADORA2A (0.46) NQO2ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5022748 0.86 ACVR1 (0.40) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5521214 0.86 ACVR1 (0.40) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5022740 0.86 ACVR1 (0.40) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL5521204 0.86 ACVR1 (0.40) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL27597784 0.84 MTOR (0.41) CCNE2CDK4CCND1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474145-B1 QUINOLINE DERIVATIVES AS NPY ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-04-23 EP claimed