SCHEMBL5085236

SCHEMBL5085236

Cc1cscc1-c1ccc(-c2cccc(Cl)c2Cl)nn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.52
CNR1 P21554 2/20 0.52
IDO1 P14902 1/20 0.41
CYP2A6 P11509 2/20 0.40
CYP2B6 P20813 2/20 0.40
NUDT1 P36639 1/20 0.38
P2RX7 Q99572 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NOTUM Q6P988 1/20 0.37
KDM1A O60341 1/20 0.37
PTPN1 P18031 1/20 0.36
MAOA P21397 1/20 0.36
MAPK1 P28482 1/20 0.36
ADRA1A P35348 1/20 0.36
SCN4A P35499 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14568111 0.76 CNR2 (0.50) CNR2CNR1IDO1NUDT1P2RX7
SCHEMBL14567764 0.75 CNR2 (0.49) CNR2CNR1IDO1CYP2A6CYP2B6
SCHEMBL5084514 0.74 CNR2 (0.57) CNR2CNR1IDO1NUDT1P2RX7
SCHEMBL5085230 0.74 CNR2 (0.48) CNR2CNR1IDO1NUDT1P2RX7
SCHEMBL14051355 0.72 CNR2 (0.52) CNR2CNR1IDO1P2RX7CYP2D6
SCHEMBL5085295 0.71 CNR2 (0.54) CNR2CNR1IDO1NUDT1P2RX7
SCHEMBL5087450 0.71 CNR2 (0.54) CNR2CNR1IDO1NUDT1P2RX7
SCHEMBL14051391 0.70 CNR2 (0.49) CNR2CNR1IDO1
SCHEMBL1764977 0.69 HTR2C (0.47) CNR2CNR1IDO1NUDT1MAPK1
SCHEMBL14051353 0.69 CNR2 (0.52) CNR2CNR1IDO1NUDT1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008116816-A1 COMBINATION OF CB2 LIGAND AND PARACETAMOL GLAXO GROUP LIMITED (GB) 2008-10-02 WO disclosed
WO-2008116816-A1 COMBINATION OF CB2 LIGAND AND PARACETAMOL GLAXO GROUP LIMITED (GB) 2008-10-02 WO disclosed
WO-2007022938-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2007-03-01 WO disclosed
WO-2007022938-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2007-03-01 WO disclosed