SCHEMBL5116828

SCHEMBL5116828

CC(Oc1ccc(CC2c3ccc(O)cc3CCN2C2CCOCC2)cc1)C1CCCCN1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.37
ESR2 Q92731 8/20 0.37
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5114923 0.94 ESR1 (0.40) ESR1ESR2KDM4EALDH1A1ALOX15
SCHEMBL5109391 0.94 ESR1 (0.39) ESR1ESR2KDM4EALDH1A1ALOX15
SCHEMBL5108109 0.91 SLC6A2 (0.37) KDM4EDRD2DRD1
Trifluoroacetic Acid SCHEMBL5113788 0.88 ESR1 (0.37) ESR1ESR2
Trifluoroacetic Acid SCHEMBL5108850 0.87 ESR1 (0.36) ESR1ESR2
SCHEMBL5115565 0.86 KDM4E (0.48) ESR1ESR2KDM4EALDH1A1ALOX15
SCHEMBL5108015 0.85 ESR1 (0.40) ESR1ESR2KDM4EALDH1A1ALOX15
SCHEMBL5102997 0.85 SLC6A2 (0.40) KDM4EDRD2DRD1
SCHEMBL5102395 0.84 SLC6A2 (0.39) KDM4EDRD2DRD1
SCHEMBL5101665 0.83 ESR1 (0.59) ESR1ESR2KDM4EALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435729-B2 Compounds and methods for modulation of estrogen receptors SIGNAL PHARMACEUTICALS, LLC (US) 2008-10-14 US disclosed