SCHEMBL5132151

SCHEMBL5132151

N#Cc1ccc2c(c1)ncc(=O)n2CCN1CC[CH]CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN7A Q01118 2/20 0.46
SCN5A Q14524 1/20 0.46
SCN2A Q99250 1/20 0.46
SCN8A Q9UQD0 1/20 0.46
KCNH2 Q12809 13/20 0.46
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL706122 0.85 KCNH2 (0.50) SCN7ASCN5ASCN2ASCN8AKCNH2
SCHEMBL923527 0.80 KCNH2 (0.51) KCNH2
SCHEMBL706674 0.79 KCNH2 (0.45) SCN7ASCN5ASCN2ASCN8AKCNH2
SCHEMBL4779522 0.78 SCN7A (0.58) SCN7ASCN5ASCN2ASCN8AKCNH2
SCHEMBL4777392 0.77 KCNH2 (0.38) KCNH2
SCHEMBL708368 0.76 KCNH2 (0.56) KCNH2CYP3A4CYP2D6
SCHEMBL12002208 0.75 KCNH2 (0.55) KCNH2CYP3A4CYP2D6
SCHEMBL4776915 0.75 KCNH2 (0.47) KCNH2
SCHEMBL922035 0.72 KCNH2 (0.57) KCNH2CYP3A4CYP2D6
SCHEMBL708597 0.71 KCNH2 (0.51) KCNH2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893599-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS AstraZeneca AB (SE) 2008-03-05 EP disclosed
WO-2006134378-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2006-12-21 WO disclosed