SCHEMBL5133145

SCHEMBL5133145

COc1ccc(OC)c(Cc2nc3c([AsH2])ncnc3n2CCC=C(C)C)c1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 11/20 0.57
HSP90AA1 P07900 10/20 0.57
ERBB2 P04626 7/20 0.57
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
HSP90B1 P14625 1/20 0.35
KCNH2 Q12809 1/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1967170 0.89 HSP90AB1 (0.73) HSP90AB1HSP90AA1ERBB2HSP90B1
SCHEMBL5416164 0.83 HSP90AB1 (0.51) HSP90AB1HSP90AA1ERBB2LMNATP53
SCHEMBL14466177 0.79 HSP90AA1 (0.59) HSP90AB1HSP90AA1ERBB2HSP90B1
SCHEMBL1965605 0.79 ERBB2 (0.73) HSP90AB1HSP90AA1ERBB2
SCHEMBL1963778 0.79 HSP90AB1 (0.73) HSP90AB1HSP90AA1ERBB2
SCHEMBL1964104 0.79 ERBB2 (0.73) HSP90AB1HSP90AA1ERBB2HSP90B1
SCHEMBL1964988 0.75 HSP90AA1 (0.78) HSP90AB1HSP90AA1ERBB2
SCHEMBL1964201 0.73 HSP90AA1 (1.00) HSP90AB1HSP90AA1ERBB2HSP90B1
SCHEMBL30583202 0.73 HSP90AA1 (1.00) HSP90AB1HSP90AA1ERBB2HSP90B1
SCHEMBL1966909 0.72 HSP90AB1 (0.80) HSP90AB1HSP90AA1ERBB2HSP90B1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962863-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 Conforma Therapeutics Corporation (US) 2008-09-03 EP disclosed
WO-2007075572-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 CONFORMA THERAPEUTICS CORPORATION (US) 2007-07-05 WO disclosed