SCHEMBL5133273

SCHEMBL5133273

COC(=O)[C@@H](C)N(CCC[AsH2])C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 2/20 0.34
CA12 O43570 1/20 0.33
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3838124 0.85 CA14 (0.34) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL2253762 0.85 CA14 (0.34) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL2253766 0.85 CA14 (0.34) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL27612964 0.85 CA14 (0.34) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL22137615 0.84 CA14 (0.39) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL19663961 0.83 CA14 (0.40) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL2153085 0.82 CA14 (0.35) CA14CA12
SCHEMBL29023150 0.82 CA14 (0.35) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL708096 0.80 CA14 (0.37) CA14CA12HDAC1HDAC2HDAC6
SCHEMBL708097 0.80 CA14 (0.37) CA14CA12HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556362-B1 BETA-AMINO HETEROCYCLIC DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO INC (US) 2008-03-26 EP disclosed