SCHEMBL5133376

SCHEMBL5133376

O=C1NCc2c(Cl)ccc(-c3cc4cc(CN5CCN(c6ccncc6)CC5)ccc4[nH]3)c21

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 17/20 0.44
TNKS O95271 1/20 0.38
PARP1 P09874 1/20 0.38
PARP10 Q53GL7 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
PARP4 Q9UKK3 1/20 0.38
PARP3 Q9Y6F1 1/20 0.38
AURKA O14965 1/20 0.38
CDK1 P06493 1/20 0.38
KDR P35968 1/20 0.38
SLC2A1 P11166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3044841 0.88 MEN1 (0.44) CHEK1PARP1PARP2AURKAKDR
Hydrochloric Acid SCHEMBL3046777 0.86 CHEK1 (0.52) CHEK1AURKACDK1KDR
Hydrochloric Acid SCHEMBL3043640 0.86 AURKA (0.44) CHEK1AURKACDK1KDR
Hydrochloric Acid SCHEMBL3033516 0.86 CHEK1 (0.50) CHEK1AURKACDK1KDR
SCHEMBL3049632 0.86 DRD4 (0.46) CHEK1PARP1AURKAKDR
Hydrochloric Acid SCHEMBL3050165 0.86 CHEK1 (0.54) CHEK1AURKAKDR
Hydrochloric Acid SCHEMBL3043804 0.85 CHEK1 (0.44) CHEK1AURKACDK1KDR
SCHEMBL3049431 0.85 CHEK1 (0.44) CHEK1AURKACDK1KDR
Hydrochloric Acid SCHEMBL3044456 0.85 CHEK1 (0.44) CHEK1AURKACDK1KDR
Hydrochloric Acid SCHEMBL3049651 0.84 CHEK1 (0.42) CHEK1PARP1PARP2AURKACDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed