SCHEMBL5134096

SCHEMBL5134096

CCCCCNCCn1c(Sc2cc(OC)ccc2I)nc2c(N)ncnc21

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 11/20 0.79
HSP90AB1 P08238 9/20 0.77
HSP90AA1 P07900 9/20 0.70
HSP90B1 P14625 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035551 0.97 ERBB2 (0.80) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5045305 0.96 ERBB2 (0.77) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5035515 0.94 ERBB2 (0.82) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5133123 0.92 ERBB2 (0.79) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL1963694 0.90 ERBB2 (0.81) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5045791 0.90 ERBB2 (0.82) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5045346 0.90 ERBB2 (0.81) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5043343 0.90 ERBB2 (0.81) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5517643 0.89 ERBB2 (0.87) ERBB2HSP90AB1HSP90AA1HSP90B1
SCHEMBL5516345 0.88 ERBB2 (0.87) ERBB2HSP90AB1HSP90AA1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962863-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 Conforma Therapeutics Corporation (US) 2008-09-03 EP disclosed
WO-2007075572-A2 ORALLY ACTIVE PURINE-BASED INHIBITORS OF HEAT SHOCK PROTEIN 90 CONFORMA THERAPEUTICS CORPORATION (US) 2007-07-05 WO disclosed