SCHEMBL5134599

SCHEMBL5134599

CCCc1nn(C)c2cnc(NCCc3cnn(-c4ccccc4)c3)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 3/20 0.40
ADORA1 P30542 4/20 0.39
MKNK2 Q9HBH9 1/20 0.38
CACNA2D1 P54289 4/20 0.38
SLC6A2 P23975 2/20 0.38
ADORA2A P29274 5/20 0.37
TMIGD3 P0DMS9 3/20 0.37
ADORA2B P29275 2/20 0.37
CYP2C9 P11712 4/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
HPGD P15428 3/20 0.36
TSHR P16473 3/20 0.36
CASP1 P29466 3/20 0.36
CYP2C19 P33261 3/20 0.36
CASP7 P55210 3/20 0.36
HSD17B10 Q99714 3/20 0.36
USP2 O75604 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133695 0.79 PDE10A (0.41) CYP2C9ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL4903712 0.76 PDE5A (0.52) ADORA1ADORA2AADORA2BALDH1A1HPGD
SCHEMBL15779863 0.71 DRD4 (0.53) CYP2C9ALDH1A1HPGDHSD17B10ALOX15
SCHEMBL16373532 0.67 ATM (0.52) CYP2C9ALDH1A1HPGDNPSR1POLB
SCHEMBL17788488 0.64 HCAR2 (0.46) CYP2C9ALDH1A1HPGDNPSR1POLB
SCHEMBL15941389 0.64 DRD4 (0.54) CYP2C9ALDH1A1HPGDHSD17B10ALOX15
SCHEMBL3122462 0.64 PDE5A (0.36) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL5133805 0.64 DRD1 (0.45) CACNA2D1CYP2D6POLB
SCHEMBL20083830 0.63 DRD4 (0.53) CYP2C9ALDH1A1HPGDHSD17B10ALOX15
SCHEMBL9608917 0.63 DRD4 (0.55) CYP2C9ALDH1A1HPGDHSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO disclosed