SCHEMBL5134955

SCHEMBL5134955

CCCCC(c1cnc(-c2ccccc2)n1CCCC)N(Cc1ccccc1)Cc1cccc(C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 1/20 0.41
NPC1 O15118 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TRPM8 Q7Z2W7 7/20 0.40
MEP1B Q16820 2/20 0.38
TSHR P16473 1/20 0.37
GABRA1 P14867 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136262 0.91 TLR7 (0.41)
SCHEMBL5135283 0.89 NPC1 (0.36) LTB4R2NPC1SMN1; SMN2TRPM8
SCHEMBL5137355 0.88 TSHR (0.39) TSHR
SCHEMBL5134818 0.88 TSHR (0.39) TSHR
SCHEMBL5134753 0.87 STAT3 (0.40) LTB4R2TSHR
SCHEMBL5135309 0.86 TLR7 (0.41)
SCHEMBL5135943 0.86 C5AR1 (0.36) TSHR
SCHEMBL5134566 0.85 TSHR (0.41) LTB4R2NPC1TSHR
SCHEMBL5137583 0.84 HSP90AA1 (0.39) TSHRGABRA1
SCHEMBL5135337 0.83 TSHR (0.37) LTB4R2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed