SCHEMBL5136143

SCHEMBL5136143

O=C(c1cn(C[C@@H]2CO2)c2cc(Cl)ccc12)N1CCC2(CC1)OCc1ccccc12

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 18/20 0.76
OXTR P30559 1/20 0.59
AVPR2 P30518 1/20 0.47
CNR1 P21554 2/20 0.45
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4356225 1.00 AVPR1A (0.76) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL4363226 0.90 AVPR1A (0.69) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL13603033 0.90 AVPR1A (0.69) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL4363221 0.90 AVPR1A (0.69) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL14160208 0.89 AVPR1A (0.72) AVPR1AOXTRAVPR2CNR1CNR2
Hydrochloric Acid SCHEMBL4358769 0.88 AVPR1A (0.71) AVPR1AOXTRAVPR2CNR1CNR2
Hydrochloric Acid SCHEMBL5137451 0.88 AVPR1A (0.71) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL4356439 0.88 AVPR1A (0.75) AVPR1AOXTRAVPR2CNR1CNR2
SCHEMBL4360998 0.87 AVPR1A (0.65) AVPR1AOXTRAVPR2CNR1
SCHEMBL5136915 0.87 AVPR1A (0.65) AVPR1AOXTRAVPR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904477-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed