SCHEMBL5136273

SCHEMBL5136273

CC(C)Oc1ccc(-c2[nH]c3nccnc3c2CN(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 19/20 0.53
GSK3B P49841 19/20 0.53
CDK1 P06493 18/20 0.53
CCNB2 O95067 17/20 0.53
CCNB1 P14635 17/20 0.53
CCNB3 Q8WWL7 17/20 0.53
CDK5 Q00535 12/20 0.53
CDK5R1 Q15078 11/20 0.53
CDK2 P24941 3/20 0.51
CCNE1 P24864 2/20 0.51
ZAP70 P43403 1/20 0.51
PTK2B Q14289 1/20 0.51
MAPK8 P45983 3/20 0.45
AURKA O14965 2/20 0.45
MAP4K4 O95819 2/20 0.45
PAK4 O96013 2/20 0.45
ABL1 P00519 2/20 0.45
FYN P06241 2/20 0.45
RET P07949 2/20 0.45
KDR P35968 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL1778365 0.82 GSK3A (0.52) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1779243 0.81 GSK3A (0.61) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL5618955 0.81 MAPK14 (0.53) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777880 0.80 GSK3A (0.65) GSK3AGSK3BCDK1CCNB2CCNB1
Iodide SCHEMBL3224491 0.80 GSK3A (0.56) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777706 0.79 GSK3A (0.55) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777025 0.79 GSK3A (0.55) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1777538 0.78 GSK3A (0.53) GSK3AGSK3BCDK1CCNB2CCNB1
Aloisine SCHEMBL79714 0.68 GSK3A (1.00) GSK3AGSK3BCDK1CCNB2CCNB1
Iodide SCHEMBL1779435 0.68 GSK3A (0.69) GSK3AGSK3BCDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1990343-A2 Azaindoles Aventis Pharma Limited (GB) 2008-11-12 EP disclosed