SCHEMBL5136333

SCHEMBL5136333

COc1ccc(C(c2cccnc2)N(c2cccnc2)c2cccnc2N)cn1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.37
CYP19A1 P11511 1/20 0.34
PFKFB3 Q16875 1/20 0.34
PDE4D Q08499 2/20 0.33
PIK3CA P42336 3/20 0.31
PIK3CD O00329 2/20 0.31
PIK3CB P42338 2/20 0.31
PIK3CG P48736 2/20 0.31
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MTOR P42345 1/20 0.31
MEN1 O00255 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469601 0.88 KCNA5 (0.42) KCNA5CYP19A1PFKFB3PDE4DKMT2A
SCHEMBL4457212 0.83 KCNA5 (0.42) KCNA5CYP19A1PDE4DKMT2AALDH1A1
SCHEMBL4461880 0.81 KCNA5 (0.35) KCNA5CYP19A1PFKFB3PDE4DPIK3CA
SCHEMBL4461835 0.80 CYP19A1 (0.40) KCNA5CYP19A1PDE4DKMT2AALDH1A1
SCHEMBL4457667 0.79 KMT2A (0.39) KCNA5CYP19A1KMT2AALDH1A1POLB
SCHEMBL4454542 0.78 CYP19A1 (0.45) KCNA5CYP19A1KMT2AMEN1
SCHEMBL4472869 0.78 CYP19A1 (0.48) KCNA5CYP19A1PFKFB3
SCHEMBL4470602 0.77 KCNA5 (0.35) KCNA5CYP19A1PFKFB3PDE4DKMT2A
SCHEMBL4468118 0.76 KCNA5 (0.36) KCNA5CYP19A1PDE4DKMT2AALDH1A1
SCHEMBL4472165 0.76 CYP19A1 (0.45) KCNA5CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981507-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-10-22 EP disclosed
WO-2007089679-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO disclosed