SCHEMBL5139624

SCHEMBL5139624

CN(CCN1CCCC1)c1ccc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)cn1.Cc1cc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)ccc1OCCN1CCC(CC(=O)O)CC1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.55
CHRM1 P11229 4/20 0.55
HTR2A P28223 3/20 0.49
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4518292 0.89 MCHR1 (0.65) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5139623 0.87 MCHR1 (0.55) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL13920416 0.82 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2321296 0.81 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2319487 0.80 MCHR1 (0.73) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2322440 0.80 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2328524 0.80 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2322150 0.80 MCHR1 (0.64) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4519229 0.79 MCHR1 (0.67) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2320676 0.79 MCHR1 (0.71) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7452911-B2 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2008-11-18 US disclosed