SCHEMBL5139729

SCHEMBL5139729

O=C(Nc1ccccc1[AsH2])c1ccc(C(C(=O)Nc2ccccc2)C(=O)Nc2cccc(F)c2)cc1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.73
HDAC3 O15379 6/20 0.60
HDAC2 Q92769 5/20 0.60
NPC1 O15118 1/20 0.54
HPGD P15428 1/20 0.54
RAB9A P51151 1/20 0.54
KCNK3 O14649 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM4E B2RXH2 1/20 0.47
KCNK9 Q9NPC2 1/20 0.47
NCOR2 Q9Y618 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689337 0.87 HDAC1 (0.96) HDAC1HDAC3HDAC2NCOR2
SCHEMBL2109226 0.84 HDAC1 (1.00) HDAC1HDAC3HDAC2NPC1HPGD
SCHEMBL2108547 0.77 HDAC1 (0.76) HDAC1HDAC3HDAC2NCOR2
SCHEMBL1754325 0.75 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR2
SCHEMBL2109945 0.74 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR2
SCHEMBL1689389 0.73 HDAC1 (0.67) HDAC1HDAC3HDAC2
SCHEMBL23447715 0.72 NPC1 (1.00) NPC1HPGDRAB9AKCNK3MEN1
SCHEMBL2108411 0.72 HDAC1 (0.74) HDAC1HDAC3HDAC2
SCHEMBL2108136 0.72 HDAC1 (0.96) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL1689351 0.72 HDAC1 (0.96) HDAC1HDAC3HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed