SCHEMBL5140274

SCHEMBL5140274

CC(C)=CCCCn1c(-c2ccccc2OCc2ccccc2)nc(C)c(-c2cc(C)cs2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 7/20 0.39
NR1I2 O75469 4/20 0.39
PTGER1 P34995 6/20 0.37
PTGER4 P35408 6/20 0.37
PTGER3 P43115 6/20 0.37
PTGER2 P43116 6/20 0.37
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
TBXA2R P21731 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
PTGFR P43088 1/20 0.36
PTGIR P43119 1/20 0.36
MAOB P27338 1/20 0.36
BRD4 O60885 1/20 0.36
DHODH Q02127 1/20 0.36
KDM4E B2RXH2 1/20 0.35
STAT3 P40763 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135738 0.86 CASR (0.49) CASRNR1I2PTGER1PTGER4PTGER3
SCHEMBL3345165 0.75 CASR (0.56) CASRNR1I2
SCHEMBL4139286 0.74 CASR (0.66) CASRNR1I2
SCHEMBL4138510 0.72 CASR (0.67) CASRNR1I2PTGER1PTGER4PTGER3
SCHEMBL4147810 0.72 CASR (0.56) CASRNR1I2BRD4
SCHEMBL4135676 0.72 CASR (0.47) CASRNR1I2PTGER1PTGER4PTGER3
SCHEMBL27751255 0.71 CASR (0.51) CASRNR1I2
SCHEMBL4144136 0.71 CASR (0.51) CASRNR1I2BRD4
SCHEMBL4142850 0.71 NR1I2 (0.70) CASRNR1I2PTGER1PTGER4PTGER3
SCHEMBL4138096 0.70 CASR (0.69) CASRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951244-A2 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP disclosed
WO-2007062370-A2 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO disclosed