SCHEMBL5140908

SCHEMBL5140908

FC(F)(F)c1ccc(C(F)(F)CN2CCC(Nc3nccc4[nH]ncc34)CC2)cc1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 20/20 0.74
KCNH2 Q12809 8/20 0.74
CYP2D6 P10635 5/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5141039 0.92 GRIN2B (0.63) GRIN2BKCNH2CYP2D6
SCHEMBL5141661 0.89 GRIN2B (0.59) GRIN2BKCNH2CYP2D6
SCHEMBL5167369 0.88 GRIN2B (0.59) GRIN2BKCNH2CYP2D6
SCHEMBL4310737 0.85 GRIN2B (1.00) GRIN2BKCNH2CYP2D6
SCHEMBL4313459 0.82 GRIN2B (0.92) GRIN2BKCNH2CYP2D6
SCHEMBL4447587 0.82 GRIN2B (0.92) GRIN2BKCNH2CYP2D6
SCHEMBL4445950 0.82 GRIN2B (0.92) GRIN2BKCNH2CYP2D6
SCHEMBL5141563 0.81 GRIN2B (0.54) GRIN2BKCNH2CYP2D6
SCHEMBL4311365 0.78 GRIN2B (0.86) GRIN2BKCNH2CYP2D6
SCHEMBL4306119 0.78 GRIN2B (0.85) GRIN2BKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874318-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006113471-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2006-10-26 WO disclosed