SCHEMBL5148290

SCHEMBL5148290

O=C(c1ccco1)C1CNCCN1c1cc(N2CCOCC2)nc(-n2c(CO)nc3ccccc32)n1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 3/20 0.44
CD274 Q9NZQ7 3/20 0.44
ATR Q13535 3/20 0.44
CHEK1 O14757 2/20 0.44
ATRIP Q8WXE1 2/20 0.44
PIK3CB P42338 14/20 0.43
PIK3CD O00329 9/20 0.41
PIK3CA P42336 8/20 0.41
PIK3CG P48736 4/20 0.40
PIK3R1 P27986 1/20 0.40
GBA1 P04062 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700323 0.92 PIK3CB (0.48) PIK3CBPIK3CDPIK3CAPIK3CGPIK3R1
SCHEMBL2954006 0.81 PIK3CB (0.49) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL3696106 0.79 PIK3CB (0.65) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL2954762 0.74 PIK3CB (0.60) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL2956597 0.74 PIK3CB (0.56) PIK3CBPIK3CDPIK3CAPIK3CGPIK3R1
SCHEMBL2955577 0.73 PIK3CB (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL2954585 0.73 PIK3CB (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL2947721 0.72 PIK3CB (0.52) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL373245 0.72 PDCD1 (0.56) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL2948267 0.72 PIK3CB (0.52) PDCD1CD274ATRCHEK1ATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1864665-A1 IMMUNOSUPPRESSIVE AGENT AND ANTI-TUMOR AGENT COMPRISING HETEROCYCLIC COMPOUND AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2007-12-12 EP claimed
EP-1864665-A1 IMMUNOSUPPRESSIVE AGENT AND ANTI-TUMOR AGENT COMPRISING HETEROCYCLIC COMPOUND AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2007-12-12 EP disclosed