SCHEMBL5151129

SCHEMBL5151129

Cc1cc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)ccc1OCCNC(CO)CO

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.59
CHRM1 P11229 4/20 0.59
HTR2A P28223 3/20 0.43
CYP2D6 P10635 1/20 0.43
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
ACACB O00763 2/20 0.38
HTR1A P08908 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2319440 0.87 MCHR1 (0.68) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL5155090 0.85 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4477045 0.84 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4474578 0.84 MCHR1 (0.60) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4486672 0.83 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4469369 0.83 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4475254 0.83 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4475563 0.82 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4477315 0.82 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL5158521 0.81 MCHR1 (0.55) MCHR1CHRM1HTR2ACYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740572-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-10 EP disclosed
WO-2005103031-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed