SCHEMBL5154531

SCHEMBL5154531

CC1OCC[C]C1Cc1ccc(C#Cc2ccc3cc(-c4ccc(Cl)cc4)ccc3n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.35
CHRM1 P11229 1/20 0.35
HTR2A P28223 1/20 0.35
BACE1 P56817 1/20 0.34
GRM5 P41594 1/20 0.31
TTR P02766 1/20 0.31
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5155292 0.73 NPC1 (0.39) MCHR1CHRM1HTR2ABACE1ACACB
SCHEMBL2325485 0.72 MCHR1 (0.54) MCHR1CHRM1HTR2ABACE1
SCHEMBL6381920 0.71 MCHR1 (0.39) MCHR1CHRM1HTR2ABACE1
SCHEMBL2322808 0.68 BACE1 (0.46) MCHR1CHRM1HTR2ABACE1GRM5
SCHEMBL2322357 0.64 MCHR1 (0.71) MCHR1CHRM1HTR2A
SCHEMBL2328403 0.62 NPC1 (0.46) MCHR1CHRM1HTR2A
SCHEMBL2321084 0.58 MCHR1 (0.58) MCHR1CHRM1HTR2ABACE1
SCHEMBL12884284 0.58 TTR (0.56) BACE1GRM5TTR
SCHEMBL28255967 0.56 BACE1 (0.63) MCHR1BACE1
SCHEMBL4480442 0.56 MCHR1 (0.78) MCHR1CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740572-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-10 EP claimed
WO-2005103031-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO claimed