SCHEMBL5155035

SCHEMBL5155035

C[C@@]1(O)CCN(CCc2ccc(C#Cc3ccc(-c4ccc(Cl)cc4)cn3)cc2)C[C@@H]1O

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 18/20 0.66
CHRM1 P11229 4/20 0.51
HTR2A P28223 3/20 0.51
CYP2D6 P10635 1/20 0.50
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ACACB O00763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492516 0.88 MCHR1 (0.76) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4493322 0.86 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5154904 0.81 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6385251 0.81 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2325467 0.80 MCHR1 (1.00) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4480442 0.80 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6380398 0.78 MCHR1 (0.46) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5151568 0.78 MCHR1 (0.68) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4478438 0.77 MCHR1 (0.77) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4484488 0.77 MCHR1 (0.77) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740572-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-10 EP disclosed
WO-2005103031-A1 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed