SCHEMBL5159484

SCHEMBL5159484

O=C(NC(=O)C1CCOCC1)c1ncccc1NC(=O)c1cccc2ccccc12

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 13/20 0.71
CNR2 P34972 11/20 0.71
KDM4E B2RXH2 2/20 0.56
MAPT P10636 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CYP2C9 P11712 2/20 0.49
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.46
CYP3A4 P08684 1/20 0.46
KDR P35968 1/20 0.44
BACE1 P56817 1/20 0.44
ULK1 O75385 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5163296 0.86 CNR1 (0.54) CNR1CNR2SMN1; SMN2CYP2C9NPC1
SCHEMBL5236479 0.85 CNR1 (0.73) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5164108 0.83 CNR1 (1.00) CNR1CNR2CYP2C9ALDH1A1NPC1
SCHEMBL5236769 0.80 CNR1 (0.66) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5230358 0.78 CNR1 (0.72) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5232573 0.78 CNR1 (0.70) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5238904 0.77 CNR1 (0.72) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5238111 0.77 CNR1 (0.69) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5236233 0.75 CNR1 (0.67) CNR1CNR2KDM4EMAPTSMN1; SMN2
SCHEMBL5235653 0.75 CNR1 (0.71) CNR1CNR2KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756061-A1 THERAPEUTIC COMPOUNDS: PYRIDINE N OXIDE SCAFFOLD AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115987-A1 THERAPEUTIC COMPOUNDS: PYRIDINE N OXIDE SCAFFOLD ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756061-A1 THERAPEUTIC COMPOUNDS: PYRIDINE N OXIDE SCAFFOLD AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115987-A1 THERAPEUTIC COMPOUNDS: PYRIDINE N OXIDE SCAFFOLD ASTRAZENECA AB (SE) 2005-12-08 WO disclosed