SCHEMBL516614

SCHEMBL516614

NS(=O)(=O)c1ccc2cc[nH]c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.60
CA2 P00918 3/20 0.60
CA12 O43570 2/20 0.60
CA9 Q16790 1/20 0.60
HTR6 P50406 1/20 0.53
LMNA P02545 1/20 0.50
ESR1 P03372 5/20 0.49
CYP19A1 P11511 1/20 0.49
CYP2A6 P11509 1/20 0.47
AHR P35869 3/20 0.47
CMA1 P23946 1/20 0.47
TYR P14679 1/20 0.47
ENPP2 Q13822 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CDK8 P49336 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31497301 1.00 CA1 (0.60) CA1CA2CA12CA9HTR6
Hydrochloric Acid SCHEMBL5241443 0.98 CA1 (0.58) CA1CA2CA12CA9HTR6
SCHEMBL516725 0.85 CA1 (0.75) CA1CA2CA12CA9LMNA
Hydrochloric Acid SCHEMBL19211662 0.83 CA1 (0.73) CA1CA2CA12CA9LMNA
SCHEMBL7137662 0.82 MEN1 (0.66) CA1CA2HTR6ESR1CYP19A1
SCHEMBL1035779 0.81 ESR1 (0.53) CA1CA2CA12CA9HTR6
SCHEMBL1144770 0.81 ESR1 (0.53) CA1CA2CA12CA9HTR6
SCHEMBL1120379 0.81 TYR (0.52) CA1CA2CA12CA9HTR6
SCHEMBL30260844 0.81 ESR1 (0.53) CA1CA2CA12CA9HTR6
Hydrochloric Acid SCHEMBL28101627 0.79 TYR (0.50) CA1CA2CA12CA9HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 102 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105272904-B N- phenylamide compound and its application 中国科学院广州生物医药与健康研究院 2019-04-09 CN claimed
CN-104530014-B Sulfamide compound of the dihydrobenzo of 2 oxo 1,2 [cd] indoles 6 and combinations thereof and application 中国科学院广州生物医药与健康研究院 2018-03-20 CN claimed
EP-3233845-A1 PARG INHIBITORY COMPOUNDS Cancer Research Technology Limited (GB) 2017-10-25 EP claimed
CN-107295799-A Parg inhibiting compounds 癌症研究科技有限公司 2017-10-24 CN claimed
CN-105985282-A 2-oxo-1, 2-dihydrobenzo [ cd ] indole compound and application thereof 中国科学院广州生物医药与健康研究院 2016-10-05 CN claimed
WO-2016097749-A1 PARG INHIBITORY COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-06-23 WO claimed
CN-105272904-A N-phenylamide compound and application thereof GUANGZHOU INST BIOMED & HEALTH 2016-01-27 CN claimed
CN-104530014-A 2-oxo-1,2-dihydrobenzo[cd] indole-6-sulfamide compound and composition and application thereof GUANGZHOU INST BIOMED & HEALTH 2015-04-22 CN claimed
EP-2523559-A1 COMPOUNDS AND METHODS GlaxoSmithKline LLC (US) 2012-11-21 EP claimed
CN-101044114-B Nitrobenzindoles and their use in cancer therapy AUCKLAND UNISERVICES LTD. (NZ) 2012-02-15 CN claimed
WO-2011088027-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-07-21 WO claimed
EP-1869010-A1 3-SULFONYLAMINO-PYRROLIDINE-2-ONE DERIVATIVES AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2007-12-26 EP claimed
CN-101044114-A Nitrobenzindoles and their use in cancer therapy AUCKLAND UNISERVICES LTD (NZ) 2007-09-26 CN claimed
EP-1786770-A1 N-(1-(2,3-DIHYDRO-1H-INDEN-5YL) -2-OXO-3-PYRROLIDINYL) -SULFONAMIDE DERIVATIVES FOR USE AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2007-05-23 EP claimed
WO-2006108709-A1 3-SULFONYLAMINO-PYRROLIDINE-2-ONE DERIVATIVES AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2006-10-19 WO claimed
WO-2006027186-A1 N-(1-(2,3-DIHYDRO-1H-INDEN-5YL) -2-OXO-3-PYRROLIDINYL) -SULFONAMIDE DERIVATIVES FOR USE AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
CN-1162596-A Antiarrhythmic Agents AMERICAN CYANAMID CO (US) 1997-10-22 CN claimed
EP-0230035-B1 Omega-[(hetero)alkyl]benz[cd]indol-2-amines AMERICAN CYANAMID CO (US) 1994-10-12 EP claimed
CN-119798210-B Preparation method of high-purity glycolide 山东金特安全科技有限公司 2025-05-20 CN disclosed
US-4615966-A Color transfer photographic processes and products with indole phthalein filter dyes POLAROID CORPORATION (US) 1986-10-07 US disclosed