SCHEMBL5166696

SCHEMBL5166696

CC1(c2ccc(Br)cc2)COC1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
CYP3A4 P08684 1/20 0.39
KCNH2 Q12809 1/20 0.37
OPRM1 P35372 3/20 0.33
OPRD1 P41143 3/20 0.33
OPRK1 P41145 3/20 0.33
DRD1 P21728 2/20 0.33
RORC P51449 2/20 0.33
OPRL1 P41146 2/20 0.33
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
HSD11B1 P28845 1/20 0.32
ALDH1A1 P00352 2/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM1A O60341 1/20 0.30
RCOR1 Q9UKL0 1/20 0.30
HSD17B10 Q99714 1/20 0.30
G6PD P11413 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13473 0.84 TAAR1 (0.50) TAAR1KCNH2RORCALDH1A1HSD17B10
SCHEMBL13471 0.76 KCNH2 (0.44) KCNH2OPRM1OPRK1OPRL1ALDH1A1
SCHEMBL2462689 0.72 TDP1 (0.67) TDP1CYP3A4ESR1ESR2ALDH1A1
SCHEMBL739399 0.72 TDP1 (0.67) TDP1CYP3A4ESR1ESR2ALDH1A1
Hydrogen Sulfide SCHEMBL27986656 0.70 TDP1 (0.63) TDP1CYP3A4ESR1ESR2ALDH1A1
Water SCHEMBL27986199 0.70 TDP1 (0.63) TDP1CYP3A4ESR1ESR2ALDH1A1
SCHEMBL3647973 0.67 CHRNA1 (0.48) KCNH2OPRD1HSD11B1ALDH1A1MAPK1
SCHEMBL11309365 0.67 CA4 (0.48) TDP1CYP3A4ESR1ESR2MAPK1
SCHEMBL13351707 0.67 KCNH2 (0.47) TDP1KCNH2
SCHEMBL5211296 0.66 TAAR1 (0.43) TAAR1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768975-A2 PYRIDYL PIPERAZINES FOR THE TREATMENT OF CNS DISORDERS Pfizer Products Inc. (US) 2007-04-04 EP disclosed
WO-2006000912-A2 PYRIDYL PIPERAZINES FOR THE TREATMENT OF CNS DISORDERS PFIZER PRODUCTS INC. (US) 2006-01-05 WO disclosed