SCHEMBL5169528

SCHEMBL5169528

CC(=O)c1ccc(Nc2ncc(I)c(NC(CO)C(C)C)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.45
FLT3 P36888 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CDK1 P06493 11/20 0.42
KDR P35968 9/20 0.42
CDK2 P24941 8/20 0.42
CA2 P00918 3/20 0.42
CDK4 P11802 2/20 0.42
CDK7 P50613 2/20 0.42
CDK9 P50750 2/20 0.42
CCNT1 O60563 1/20 0.42
CCND1 P24385 1/20 0.42
CCNH P51946 1/20 0.42
CCNB1 P14635 2/20 0.41
CCNE1 P24864 2/20 0.41
AURKA O14965 2/20 0.41
SYK P43405 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016880 1.00 CHEK1 (0.45) CHEK1FLT3NPC1RAB9ACDK1
SCHEMBL13648454 0.88 NPC1 (0.48) CHEK1FLT3NPC1RAB9ACDK1
SCHEMBL13648652 0.87 CDK1 (0.57) CHEK1CDK1KDRCDK2CA2
SCHEMBL5173644 0.87 AURKA (0.52) CHEK1FLT3NPC1RAB9ACDK1
SCHEMBL13648525 0.87 CDK1 (0.57) CHEK1CDK1KDRCDK2CA2
SCHEMBL4018345 0.87 AURKA (0.52) CHEK1FLT3NPC1RAB9ACDK1
SCHEMBL3931675 0.83 CDK1 (0.56) CDK1KDRCDK2CA2CDK4
SCHEMBL4020087 0.83 CDK2 (0.63) RAB9ACDK1KDRCDK2CA2
SCHEMBL5174690 0.83 CDK2 (0.63) RAB9ACDK1KDRCDK2CA2
SCHEMBL4016887 0.83 CHEK1 (0.45) CHEK1FLT3NPC1RAB9ACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291624-B2 CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents BAYER SCHERING PHARMA AG (DE) 2007-11-06 US disclosed