SCHEMBL5169850

SCHEMBL5169850

COc1c(-c2ccccc2)nc2ccccc2c1C(=O)NN(C(=O)O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 20/20 0.69
CYP3A4 P08684 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4898026 0.94 TACR3 (0.79) TACR3CYP3A4
SCHEMBL5171551 0.82 TACR3 (0.70) TACR3CYP3A4
SCHEMBL4895679 0.82 TACR3 (1.00) TACR3CYP3A4
SCHEMBL3959275 0.82 TACR3 (1.00) TACR3CYP3A4
SCHEMBL4903269 0.82 TACR3 (1.00) TACR3CYP3A4
SCHEMBL4897521 0.81 TACR3 (0.88) TACR3CYP3A4
SCHEMBL4906565 0.81 TACR3 (0.88) TACR3CYP3A4
SCHEMBL5172371 0.80 TACR3 (0.62) TACR3CYP3A4
SCHEMBL4907080 0.80 TACR3 (0.86) TACR3CYP3A4
SCHEMBL8271806 0.80 TACR3 (0.86) TACR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776344-A2 QUINOLINE DERIVATIVES AS NEUROKININ RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 2007-04-25 EP claimed
WO-2006013393-A2 QUINOLINE DERIVATIVES AS NEUROKININ RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 2006-02-09 WO claimed