SCHEMBL5175779

SCHEMBL5175779

CC(C)(C)CN.COc1c(NC(=O)c2ccc(C)c(-n3cc(C(=O)O)cn3)c2)cc(C(F)(F)F)cc1NS(C)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRAF P15056 19/20 0.47
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4471665 0.95 BRAF (0.50) BRAFABL1BCR
Pivalamide SCHEMBL5175771 0.93 BRAF (0.47) BRAFABL1BCR
SCHEMBL5176650 0.89 BRAF (0.45) BRAF
SCHEMBL4477561 0.89 BRAF (0.52) BRAF
SCHEMBL5175774 0.89 BRAF (0.47) BRAFABL1BCR
SCHEMBL5177542 0.88 BRAF (0.40) BRAF
SCHEMBL5177016 0.87 BRAF (0.48) BRAF
SCHEMBL5179484 0.85 ABL1 (0.38) BRAFABL1BCR
SCHEMBL5179150 0.85 BRAF (0.46) BRAF
SCHEMBL5177001 0.84 BRAF (0.48) BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756065-A1 ANTI-CYTOKINE HETEROCYCLIC COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2007-02-28 EP disclosed
WO-2005115991-A1 ANTI-CYTOKINE HETEROCYCLIC COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-12-08 WO disclosed