SCHEMBL5178024

SCHEMBL5178024

CC(C)(C)CN.COc1c(C#N)cc(C(C)(C)C)cc1NC(=O)c1ccc(C)c(-n2cc(C(=O)O)cn2)c1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.41
MAPK14 Q16539 7/20 0.40
MAPK11 Q15759 1/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486661 0.95 MAPK14 (0.43) XDHMAPK14ABL1BCR
Pivalamide SCHEMBL5178016 0.93 MAPK14 (0.41) XDHMAPK14MAPK11ABL1BCR
SCHEMBL5179484 0.89 ABL1 (0.38) MAPK14MAPK11ABL1BCR
SCHEMBL5178018 0.89 MAPK14 (0.41) XDHMAPK14MAPK11ABL1BCR
SCHEMBL4491863 0.85 ABL1 (0.41) MAPK14MAPK11ABL1BCR
SCHEMBL5176158 0.84 MAPK14 (0.39) MAPK14
SCHEMBL4478482 0.84 ABL1 (0.41) MAPK14MAPK11ABL1BCR
SCHEMBL5176650 0.82 BRAF (0.45) MAPK14
Pivalamide SCHEMBL5179479 0.82 ABL1 (0.39) MAPK14MAPK11ABL1BCR
SCHEMBL4467266 0.82 MAPK14 (0.41) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756065-A1 ANTI-CYTOKINE HETEROCYCLIC COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2007-02-28 EP disclosed
WO-2005115991-A1 ANTI-CYTOKINE HETEROCYCLIC COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-12-08 WO disclosed