SCHEMBL5178303

SCHEMBL5178303

CCc1n[nH]cc1NC(=O)Cc1ccc(Oc2ncnc3cc(OC)c(OC)cc23)cc1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 12/20 0.70
FLT3 P36888 10/20 0.70
FLT4 P35916 9/20 0.64
CSF1R P07333 5/20 0.64
KDR P35968 10/20 0.59
CYP2C9 P11712 1/20 0.59
PDGFRA P16234 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177763 0.89 PDGFRB (0.67) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL5177825 0.89 PDGFRB (0.56) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL5177962 0.88 PDGFRB (0.72) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL5178990 0.87 PDGFRB (0.64) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL5179514 0.85 PDGFRB (0.62) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1097872 0.80 PDGFRB (0.70) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1098225 0.80 PDGFRB (0.65) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1098822 0.79 PDGFRB (0.65) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1098249 0.78 PDGFRB (1.00) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL1097832 0.78 PDGFRB (0.67) PDGFRBFLT3FLT4CSF1RKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802591-A1 QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2007-07-04 EP disclosed
WO-2006040520-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2006-04-20 WO disclosed