SCHEMBL5190835

SCHEMBL5190835

O=C(O)c1ccc2ncnc(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2c1

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 16/20 0.77
EGFR P00533 14/20 0.77
LCK P06239 1/20 0.77
AURKA O14965 1/20 0.65
RPS6KB1 P23443 1/20 0.65
ERBB3 P21860 1/20 0.62
ERBB4 Q15303 1/20 0.62
KCNH2 Q12809 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708572 0.89 ERBB2 (0.72) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL5568971 0.88 ERBB2 (0.76) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL6957615 0.88 ERBB2 (0.71) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL9973619 0.86 ERBB2 (0.73) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL30125866 0.86 ERBB2 (0.73) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL2989878 0.86 ERBB2 (0.73) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL17845956 0.86 ERBB2 (0.73) ERBB2EGFRLCKAURKARPS6KB1
SCHEMBL6980188 0.86 ERBB2 (0.73) ERBB2EGFRLCKAURKARPS6KB1
Hydrochloric Acid SCHEMBL17845945 0.85 ERBB2 (0.72) ERBB2EGFRLCKAURKARPS6KB1
Hydrochloric Acid SCHEMBL29793455 0.85 ERBB2 (0.72) ERBB2EGFRLCKAURKARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1854789-B1 QUINAZOLINE DERIVATIVE HAVING TYROSINE KINASE INHIBITORY ACTIVITY SHIONOGI & CO (JP) 2013-10-09 EP disclosed
EP-1854789-A1 QUINAZOLINE DERIVATIVE HAVING TYROSINE KINASE INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2007-11-14 EP disclosed