SCHEMBL5190849

SCHEMBL5190849

CCCS(=O)(=O)c1ccc2[nH]c(N3C(=O)N(Cc4ccncc4)C(C)(C)C3=O)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 6/20 0.41
TAS2R8 Q9NYW2 1/20 0.37
CYP2C9 P11712 4/20 0.36
CYP2C19 P33261 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 3/20 0.35
CYP2D6 P10635 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5472858 0.93 IGF1R (0.42) IGF1R
Trifluoroacetic Acid SCHEMBL5188565 0.72 IGF1R (0.43) IGF1R
SCHEMBL2938589 0.72 IGF1R (0.52) IGF1RTAS2R8
SCHEMBL4884432 0.69 IGF1R (0.58) IGF1RTAS2R8
SCHEMBL4884448 0.69 IGF1R (0.55) IGF1RTAS2R8
SCHEMBL4889027 0.67 IGF1R (0.60) IGF1RTAS2R8
SCHEMBL1108960 0.67 CYP2C9 (0.52) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL3008275 0.66 IGF1R (0.68) IGF1RTAS2R8
SCHEMBL1100753 0.66 CYP2C9 (0.51) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL13039129 0.65 IGF1R (0.67) IGF1RTAS2R8CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773828-A1 HETEROCYCLE -SUBSTITUTED CYCLIC UREA DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL USE THEREOF AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2007-04-18 EP disclosed
WO-2006010642-A1 HETEROCYCLE-SUBSTITUTED CYCLIC UREA DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL USE THEREOF AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2006-02-02 WO disclosed