SCHEMBL5193324

SCHEMBL5193324

COC(=O)c1ccc(C(=O)OC)c(Oc2ccc(C)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.56
ALDH1A1 P00352 8/20 0.51
KDM4E B2RXH2 7/20 0.51
HPGD P15428 5/20 0.51
MAPT P10636 4/20 0.51
HSD17B10 Q99714 3/20 0.51
GLA P06280 2/20 0.51
GAA P10253 2/20 0.51
ATM Q13315 2/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
USP2 O75604 1/20 0.48
MMP13 P45452 1/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29826422 1.00 TDP1 (0.56) TDP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL4506549 0.87 KDM4E (0.50) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL4521411 0.87 KDM4E (0.50) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL490297 0.86 KDM4E (0.58) TDP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL31070288 0.85 KMT2A (0.62) TDP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL31070293 0.85 MAPT (0.60) TDP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL26563278 0.83 TDP1 (0.58) TDP1ALDH1A1KDM4EHPGDMAPT
SCHEMBL472707 0.83 KMT2A (0.48) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL472705 0.82 KMT2A (0.47) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL969512 0.82 CA12 (0.50) MAPTGAAKMT2AMEN1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833825-A1 TRICYCLIC DELTA-OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2007-09-19 EP disclosed
WO-2006069277-A1 TRICYCLIC δ-OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-06-29 WO disclosed