Misonidazole

Misonidazole

SCHEMBL51943

COCC(O)Cn1ccnc1[N+](=O)[O-]

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.66
LMNA P02545 1/20 0.47
THRB P10828 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGD P15428 1/20 0.44
CA12 O43570 5/20 0.42
CA1 P00915 5/20 0.42
CA2 P00918 5/20 0.42
CA9 Q16790 5/20 0.42
MEN1 O00255 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
OPRK1 P41145 1/20 0.41
TYMP P19971 3/20 0.40
KDM4E B2RXH2 1/20 0.40
NOS1 P29475 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Misonidazole SCHEMBL2168353 0.91 KMT2A (0.56) KMT2ALMNATHRBCYP2C19HPGD
Misonidazole SCHEMBL18770100 0.89 KMT2A (0.54) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL12396375 0.87 KMT2A (0.78) KMT2ALMNATHRBCYP2C19HPGD
Misonidazole SCHEMBL2833961 0.86 KMT2A (0.51) KMT2ALMNATHRBCYP2C19HPGD
Misonidazole SCHEMBL9762481 0.86 KMT2A (0.51) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL9441423 0.85 KMT2A (0.62) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL6275185 0.85 KMT2A (0.55) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL16367290 0.84 KMT2A (0.60) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL2358150 0.84 KMT2A (0.71) KMT2ALMNATHRBCYP2C19HPGD
SCHEMBL29287184 0.84 KMT2A (0.63) KMT2ALMNATHRBCYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6585 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105121-A1 ANTICANCER FORMULATIONS AND USES THEREOF INTRAGEL THERAPEUTICS LTD. (IL) 2026-05-21 WO claimed
EP-4732908-A2 CANCER TREATMENT USING COMBINATIONS OF ERK AND RAF INHIBITORS Biomed Valley Discoveries, Inc. (US) 2026-04-29 EP claimed
EP-4687863-A1 RADIOPROTECTION BY INHIBITION OF SUPEROXIDE DISMUTASE 1 Deutsches Krebsforschungszentrum (DE) 2026-02-11 EP claimed
EP-4043017-B1 CANCER TREATMENT USING COMBINATIONS OF ERK AND RAF INHIBITORS BIOMED VALLEY DISCOVERIES INC (US) 2026-01-28 EP claimed
EP-4676551-A1 RADIATION SPACER HYDROGELS, METHODS OF FORMING, AND METHODS OF USE Clearstream Technologies Limited (IE) 2026-01-14 EP claimed
US-20250367471-A1 PERFUSION MODULATED TUMOR DOSE SCULPTING WITH SINGLE DOSE RADIOTHERAPY MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2025-12-04 US claimed
EP-4062917-B1 CANCER TREATMENTS USING COMBINATIONS OF PI3K/AKT PATHWAY AND ERK INHIBITORS BIOMED VALLEY DISCOVERIES INC (US) 2025-12-03 EP claimed
US-20250345629-A1 JOINT OPTIMIZATION OF RADIONUCLIDE AND EXTERNAL BEAM RADIOTHERAPY REFLEXION MEDICAL INC (US) 2025-11-13 US claimed
US-20250222066-A1 COMPOSITIONS AND METHODS OF TREATING, PREVENTING OR INHIBITING A FACULTATIVE ANAEROBE INFECTION UNIVERSITY OF UTAH RESEARCH FOUNDATION 2025-07-10 US claimed
EP-4547023-A2 COMPOSITIONS AND METHODS OF TREATING, PREVENTING OR INHIBITING A FACULTATIVE ANAEROBE INFECTION University of Utah Research Foundation (US) 2025-05-07 EP claimed
WO-1991013633-A1 IMPROVEMENTS RELATING TO IMMUNORADIOTHERAPY CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1991-09-19 WO claimed
US-5026694-A Antitumor agents THE BRITISH COLUMBIA CANCER FOUNDATION (CA) 1991-06-25 US claimed
US-4978332-A Reduced effect on cells distant from the site MATRIX PHARMACEUTICAL, INC. (US) 1990-12-18 US claimed
US-4921963-A Platinum complexes with one radiosensitizing ligand BRITISH COLUMBIA CANCER FOUNDATION (CA) 1990-05-01 US claimed
EP-0359347-A2 Covalently-linked complexes and methods for enhanced cytotoxicity and imaging NEORX CORPORATION (US) 1990-03-21 EP claimed
EP-0335966-A4 VASOCONSTRICTIVE SUBSTANCES IN COMBINATION WITH CYTOTOXIC AGENTS. MATRIX PHARMA INC (US) 1990-02-20 EP claimed
EP-0335966-A1 VASOCONSTRICTIVE SUBSTANCES IN COMBINATION WITH CYTOTOXIC AGENTS MATRIX PHARMACEUTICALS, INC. (US) 1989-10-11 EP claimed
EP-0330201-A2 Method of enhancing the effect of cytotoxic agents NEORX CORPORATION (US) 1989-08-30 EP claimed
WO-1989002734-A1 VASOCONSTRICTIVE SUBSTANCES IN COMBINATION WITH CYTOTOXIC AGENTS MATRIX PHARMACEUTICALS, INC. (US) 1989-04-06 WO claimed
EP-0287317-A2 Platinum complexes with one radiosensitizing ligand THE BRITISH COLUMBIA CANCER FOUNDATION (CA) 1988-10-19 EP claimed