SCHEMBL5196284

SCHEMBL5196284

NC(=O)c1cccnc1CBr

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.53
SYK P43405 3/20 0.51
KDM4E B2RXH2 6/20 0.49
ALDH1A1 P00352 4/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
NAPRT Q6XQN6 1/20 0.44
MAPT P10636 4/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
AHR P35869 1/20 0.44
P2RX7 Q99572 1/20 0.43
HTT P42858 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
BLM P54132 1/20 0.41
AGER Q15109 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497429 0.85 PARP1 (0.53) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL1937751 0.85 PARP1 (0.53) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL2108503 0.84 KDM4E (0.45) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL3664193 0.83 PARP1 (0.51) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL31439135 0.83 PARP1 (0.51) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL3967245 0.83 PARP1 (0.51) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL30011332 0.83 KDM4E (0.55) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL353231 0.83 KDM4E (0.55) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL30666151 0.83 PARP1 (0.51) PARP1SYKKDM4EALDH1A1HPGD
SCHEMBL5252687 0.82 KDM4E (0.59) KDM4EALDH1A1NAPRTMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814853-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed
WO-2006053039-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed