SCHEMBL5197278

SCHEMBL5197278

Cc1ccccc1-c1nc(-c2ccncc2)c(-c2ccc(Cl)cc2)[nH]1

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 14/20 0.70
MAPK13 O15264 13/20 0.70
MAPK12 P53778 13/20 0.70
MAPK11 Q15759 13/20 0.70
RAF1 P04049 3/20 0.70
GCGR P47871 12/20 0.68
TEK Q02763 1/20 0.65
CSNK1D P48730 1/20 0.58
CSNK1E P49674 1/20 0.58
ALOX5 P09917 2/20 0.56
MAPK9 P45984 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8791925 0.88 GCGR (0.62) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL17002223 0.87 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL5198574 0.87 MAPK14 (0.73) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL5184633 0.86 MAPK14 (0.70) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL5197475 0.85 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL8791626 0.85 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL6468726 0.84 MAPK14 (0.65) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL6468355 0.84 MAPK14 (0.78) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL6961281 0.82 MAPK14 (0.65) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL5921854 0.82 MAPK14 (0.65) MAPK14MAPK13MAPK12MAPK11RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1846389-A1 IMIDAZOLE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-10-24 EP disclosed
WO-2006082002-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-08-10 WO disclosed
US-20060173048-A1 Imidazole derivatives F. HOFFMAN-LA ROCHE AG (CH) 2006-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173048-A1 Imidazole derivatives GRM2, GRM1, GRIN2C MAPK14 2620/4885MAPK13 2722/4885MAPK12 2936/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.