SCHEMBL5198224

SCHEMBL5198224

O=C(O)[C@@H]1CC(OC(=O)[C@@H]2CC(O)CN2)CN1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.43
CYP1A2 P05177 2/20 0.43
ALOX15 P16050 2/20 0.43
CYP2C19 P33261 2/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
ARG1 P05089 1/20 0.35
DPP4 P27487 4/20 0.35
DPP8 Q6V1X1 4/20 0.35
DPP9 Q86TI2 4/20 0.35
LMNA P02545 2/20 0.33
BLM P54132 2/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.33
THRB P10828 1/20 0.33
PMP22 Q01453 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293342 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL7594974 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL2029987 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL2029661 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL2031639 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL5198220 1.00 CYP2D6 (0.43) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL11771639 0.83 DPP4 (0.33) DPP4DPP8DPP9
SCHEMBL6858335 0.82 CYP2D6 (0.60) CYP2D6CYP1A2ALOX15CYP2C19SLC1A3
SCHEMBL200243 0.82
SCHEMBL2024894 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1276491-B9 TAMANDARIN AND DIDEMNIN ANALOGS AND METHODS OF MAKING AND USING THEM UNIV PENNSYLVANIA (US) 2007-02-28 EP claimed
EP-1276491-B1 TAMANDARIN AND DIDEMNIN ANALOGS AND METHODS OF MAKING AND USING THEM UNIV PENNSYLVANIA (US) 2006-09-20 EP claimed