SCHEMBL5198546

SCHEMBL5198546

C=C(C)CC(N)c1cc(NC(=O)Cn2cc(Oc3ncnc4cc(OC)c(OC)cc34)cn2)ccc1OC

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 16/20 0.67
FLT3 P36888 14/20 0.67
FLT4 P35916 13/20 0.67
CSF1R P07333 12/20 0.67
KDR P35968 6/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4526346 0.84 PDGFRB (0.69) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4525364 0.82 PDGFRB (0.76) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4524898 0.81 PDGFRB (0.75) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4532891 0.81 PDGFRB (0.75) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4515269 0.79 PDGFRB (0.73) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4521765 0.79 PDGFRB (0.81) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4518073 0.79 PDGFRB (0.69) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4529649 0.79 PDGFRB (0.73) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4531905 0.79 PDGFRB (0.72) PDGFRBFLT3FLT4CSF1RKDR
SCHEMBL4533976 0.79 PDGFRB (0.72) PDGFRBFLT3FLT4CSF1RKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802608-A1 QUINAZOLINE DERIVATIVES FOR USE AGAINST CANCER AstraZeneca AB (SE) 2007-07-04 EP disclosed
WO-2006040526-A1 QUINAZOLINE DERIVATIVES FOR USE AGAINST CANCER ASTRAZENECA AB (SE) 2006-04-20 WO disclosed