SCHEMBL5198628

SCHEMBL5198628

Clc1ccc(-c2ccc(C#Cc3ccc([CH][C@@H]4CCCN4)cc3)nc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 18/20 0.48
CHRM1 P11229 4/20 0.47
HTR2A P28223 3/20 0.47
CYP2D6 P10635 1/20 0.47
ACACB O00763 1/20 0.36
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4493107 0.78 MCHR1 (0.51) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4493104 0.76 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6365733 0.72 MCHR1 (0.48) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL5258320 0.72 MCHR1 (0.48) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL6429354 0.71 MCHR1 (0.67) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5114893 0.71 MCHR1 (0.40) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL6365091 0.71 MCHR1 (0.52) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5154979 0.71 MCHR1 (0.52) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5228668 0.70 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL6364870 0.70 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737823-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2007-01-03 EP claimed
WO-2005103002-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO claimed